DRUGS sens assoc res assoc tot 1011 - ABT-263 [BCL2, BCL2L1, BCL2L2] 2 0 2 119 - Lapatinib [ERBB2, EGFR] 2 0 2 1268 - XAV 939 [TNKS1 (tankyrase-1)] 0 2 2 167 - OSU-03012 [PDPK1 (PDK1)] 1 1 2 204 - Tipifarnib [Farnesyl-transferase (FNTA)] 0 2 2 255 - CP724714 [ERBB2] 2 0 2 1003 - Camptothecin [TOP1] 0 1 1 1010 - Gefitinib [EGFR] 1 0 1 1020 - Lenalidomide [TNFA] 0 1 1 1030 - KU-55933 [ATM] 1 0 1 1032 - Afatinib [ERBB2, EGFR] 1 0 1 1057 - NVP-BEZ235 [PI3K (Class 1) and MTORC1/2] 0 1 1 1114 - Cetuximab [EGFR] 1 0 1 1218 - JQ1 [BRD2, BRD3, BRD4] 1 0 1 1375 - Temozolomide [DNA akylating agent] 0 1 1 1377 - Afatinib (rescreen) [ERBB2, EGFR] 1 0 1 140 - Vinorelbine [Microtubules] 0 1 1 147 - NSC-87877 [PTPN6 (SHP-1), PTPN11 (SHP-2)] 1 0 1 150 - Bicalutamide [ANDR (androgen receptor)] 1 0 1 1526 - RDEA119 (rescreen) [MAP2K1 (MEK1), MAP2K2 (MEK2)] 0 1 1 159 - HG-6-64-1 [BRAFV600E, TAK, MAP4K5] 0 1 1 170 - Shikonin [unknown] 1 0 1 180 - Thapsigargin [sarco-endoplasmic reticulum Ca2+-ATPases] 0 1 1 184 - BMS-754807 [IGF1R] 0 1 1 201 - Epothilone B [Microtubules] 0 1 1 206 - Ruxolitinib [JAK1, JAK2, TYK2] 1 0 1 224 - AS605240 [PI3Kgamma] 1 0 1 235 - QL-XII-47 [BTK, BMX] 0 1 1 275 - I-BET [BRD2, BRD3, BRD4] 1 0 1 293 - MP470 [PDGFR] 1 0 1 301 - PHA-793887 [CDK-pan] 1 0 1 306 - TG101348 [JAK2] 1 0 1 312 - AV-951 [VEGFR] 1 0 1 41 - S-Trityl-L-cysteine [KIF11] 0 1 1 53 - CGP-60474 [CDK1,CDK2,CDK5,CDK7,CDK9] 0 1 1 88 - MS-275 [HDAC] 0 1 1